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PI4K III alpha Kinase Enzyme Activity Assay Kit

The PI4K III alpha Kinase Enzyme Activity Assay Kit offers a validated, ready-to-use biochemical assay based on the renowned ADP Hunter™ Plus Assay platform from DiscoverX for accurately measuring kinase inhibitor efficacy. The kit includes recombinant PI4K III alpha, substrate, ATP, detection reagents, and assay plates, enabling precise quantification of ADP accumulation. Designed to handle elevated ATP concentrations, this assay delivers robust, reliable data ideal for high-throughput screening (HTS) and other drug discovery applications.

Biological information

Background

The Kinase Enzyme Activity Assay Kit provides a reliable biochemical method for evaluating kinase inhibitors. Built on HitHunter® assay technology, this kit is specifically optimized for PI4KIIIalpha. It comes with all essential components, including recombinant PI4KIIIalpha (Eurofins #14-908), a substrate, ATP, detection reagents, and assay plates. Each kit is accompanied by a Certificate of Analysis (COA), which outlines the recommended reaction conditions for accurate inhibitor detection. The supplied materials are sufficient to perform experiments covering two, six or twenty five 384-well assay plates.

Phosphatidylinositol 4-kinase type III alpha (PI4KIIIα, UniProt: Q9UBF8) is a lipid kinase that generates phosphatidylinositol 4-phosphate, a key precursor in the phosphoinositide signaling pathway. PI4KIIIα plays roles in Golgi function, vesicle trafficking, and viral replication. Dysregulation has been associated with cancer and viral infections, making it an attractive therapeutic target. A PI4K III alpha enzyme activity assay kit enables researchers to measure enzyme function and inhibitor effects, supporting drug discovery in oncology and antiviral research.

Target class
Kinase
Family
Type III PI4K
Accession number
GenBank NM_058004.1
Target Name
PI4K III alpha Kinase Enzyme Activity Assay Kit
Target Alias
PI4K-alpha
Origin
Human
Theori. MW
Affinity tag

Product specifications

Expression system
Purity
Purification method
Sample Buffer
Specified activity
Application
Storage conditions
1 year at -70°C
Usage disclaimer

Chemical data

Background

The Kinase Enzyme Activity Assay Kit provides a reliable biochemical method for evaluating kinase inhibitors. Built on HitHunter® assay technology, this kit is specifically optimized for PI4KIIIalpha. It comes with all essential components, including recombinant PI4KIIIalpha (Eurofins #14-908), a substrate, ATP, detection reagents, and assay plates. Each kit is accompanied by a Certificate of Analysis (COA), which outlines the recommended reaction conditions for accurate inhibitor detection. The supplied materials are sufficient to perform experiments covering two, six or twenty five 384-well assay plates.

Phosphatidylinositol 4-kinase type III alpha (PI4KIIIα, UniProt: Q9UBF8) is a lipid kinase that generates phosphatidylinositol 4-phosphate, a key precursor in the phosphoinositide signaling pathway. PI4KIIIα plays roles in Golgi function, vesicle trafficking, and viral replication. Dysregulation has been associated with cancer and viral infections, making it an attractive therapeutic target. A PI4K III alpha enzyme activity assay kit enables researchers to measure enzyme function and inhibitor effects, supporting drug discovery in oncology and antiviral research.

Compound name
Kinase
Catalog number
44-908
Molecular formula
CAS
MW
Ka
Percent composition

Product specifications

Physical state
Purity (HPLC 214nm)
Retention time (RP18 HPLC)
CMC
Exact mass
Stability
Solubility structure

Kinase Activity Assay Biological information

Background

The Kinase Enzyme Activity Assay Kit provides a reliable biochemical method for evaluating kinase inhibitors. Built on HitHunter® assay technology, this kit is specifically optimized for PI4KIIIalpha. It comes with all essential components, including recombinant PI4KIIIalpha (Eurofins #14-908), a substrate, ATP, detection reagents, and assay plates. Each kit is accompanied by a Certificate of Analysis (COA), which outlines the recommended reaction conditions for accurate inhibitor detection. The supplied materials are sufficient to perform experiments covering two, six or twenty five 384-well assay plates.

Phosphatidylinositol 4-kinase type III alpha (PI4KIIIα, UniProt: Q9UBF8) is a lipid kinase that generates phosphatidylinositol 4-phosphate, a key precursor in the phosphoinositide signaling pathway. PI4KIIIα plays roles in Golgi function, vesicle trafficking, and viral replication. Dysregulation has been associated with cancer and viral infections, making it an attractive therapeutic target. A PI4K III alpha enzyme activity assay kit enables researchers to measure enzyme function and inhibitor effects, supporting drug discovery in oncology and antiviral research.

Target class
Kinase
Family
Type III PI4K
Subfamily
PI3/PI4-kinase
Protein Name
PI4KA
Protein Alias
PI4K-alpha
Accession Number
GenBank NM_058004.1
UniProt Number
P42356
Gene Name
PI4KA
Gene ID
5297
Gene Aliases

SPG84; GIDID2; PIK4CA; PMGYCHA; pi4K230; PI4K-ALPHA

Target Species
Human

Kinase Activity Assay Usage

Product Type
Enzyme Activity Assay Kits
Application
Drug Discovery & Development
Storage Conditions
1 year at -70°C
Usage disclaimer

For Research Use Only. These products may be covered by issued US and/or foreign patents, patent applications and subject to a Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information.

Kinase Activity Assay Information

Assay Type
Enzymatic
Assay Measures
ADP Accumulation

Biological Information

Background

The Kinase Enzyme Activity Assay Kit provides a reliable biochemical method for evaluating kinase inhibitors. Built on HitHunter® assay technology, this kit is specifically optimized for PI4KIIIalpha. It comes with all essential components, including recombinant PI4KIIIalpha (Eurofins #14-908), a substrate, ATP, detection reagents, and assay plates. Each kit is accompanied by a Certificate of Analysis (COA), which outlines the recommended reaction conditions for accurate inhibitor detection. The supplied materials are sufficient to perform experiments covering two, six or twenty five 384-well assay plates.

Phosphatidylinositol 4-kinase type III alpha (PI4KIIIα, UniProt: Q9UBF8) is a lipid kinase that generates phosphatidylinositol 4-phosphate, a key precursor in the phosphoinositide signaling pathway. PI4KIIIα plays roles in Golgi function, vesicle trafficking, and viral replication. Dysregulation has been associated with cancer and viral infections, making it an attractive therapeutic target. A PI4K III alpha enzyme activity assay kit enables researchers to measure enzyme function and inhibitor effects, supporting drug discovery in oncology and antiviral research.

Target class
Kinase
Family
Type III PI4K
Accession Number
GenBank NM_058004.1
Target Name
PI4KA
Target Alias
PI4K-alpha
Origin
Human
Theoretical MW
Affinity Tag

Product Specifications

Expression system
Purity
Purification method
Sample Buffer
Enzymatic
Specified activity
Application
Drug Discovery & Development
Storage conditions
1 year at -70°C
Usage disclaimer

For Research Use Only. These products may be covered by issued US and/or foreign patents, patent applications and subject to a Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information.

Biological Information

Background

The Kinase Enzyme Activity Assay Kit provides a reliable biochemical method for evaluating kinase inhibitors. Built on HitHunter® assay technology, this kit is specifically optimized for PI4KIIIalpha. It comes with all essential components, including recombinant PI4KIIIalpha (Eurofins #14-908), a substrate, ATP, detection reagents, and assay plates. Each kit is accompanied by a Certificate of Analysis (COA), which outlines the recommended reaction conditions for accurate inhibitor detection. The supplied materials are sufficient to perform experiments covering two, six or twenty five 384-well assay plates.

Phosphatidylinositol 4-kinase type III alpha (PI4KIIIα, UniProt: Q9UBF8) is a lipid kinase that generates phosphatidylinositol 4-phosphate, a key precursor in the phosphoinositide signaling pathway. PI4KIIIα plays roles in Golgi function, vesicle trafficking, and viral replication. Dysregulation has been associated with cancer and viral infections, making it an attractive therapeutic target. A PI4K III alpha enzyme activity assay kit enables researchers to measure enzyme function and inhibitor effects, supporting drug discovery in oncology and antiviral research.

Target class
Kinase
Family
Type III PI4K
Accession Number
GenBank NM_058004.1
Target Name
PI4KA
Target Alias
PI4K-alpha
Origin
Human
Theoretical MW
Affinity Tag

Product Specifications

Expression system
Purity
Purification method
Sample Buffer
Enzymatic
Specified activity
Application
Drug Discovery & Development
Storage conditions
1 year at -70°C
Usage disclaimer

For Research Use Only. These products may be covered by issued US and/or foreign patents, patent applications and subject to a Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information.

Datasheets
44-908x Datasheet
User Manual
File N°2
Kinase Enzyme Activity Assay User Manual Rev 1
€ 1 400,00 EUR
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